Overview

Bupropion Stereoselective Disposition and CYP2D6-mediated Drug Interactions in Healthy Volunteers

Status:
Completed
Trial end date:
2019-05-01
Target enrollment:
Participant gender:
Summary
Primary objectives: 1. To comprehensively characterize steady state stereoselective pharmacokinetics of bupropion and its primary and secondary metabolites in healthy volunteers 2. To prospectively determine the time course (onset), extent and offset of CYP2D6 inhibition in relation to the pharmacokinetic profiles of bupropion and metabolites.
Phase:
Early Phase 1
Details
Lead Sponsor:
Indiana University
Collaborator:
National Institute of General Medical Sciences (NIGMS)
Treatments:
Bupropion
Dextromethorphan